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OAK 2005 Aarhus

 

 

 

PROGRAMME
Friday, June 17th

10.30-12.00

GOOD MORNING STEREOLOGY / Chaired by Bente Pakkenberg

10.30

Paul Cumming: Welcome

10.45

Jacob Jelsing:
The prefrontal cortex of the Göttingen minipig brain defined by neural projection criteria and cytoarchitecture

11.00

Anette Stark:
Neuron volume in the human neocortex

11.15

Nina Eriksen:
Neocortical cell number in the common minke whale (Balenoptera acutorostrata) brain

11.30

Katrine Fabricius:
Early induced stress and the consequences on the total neuron number in the hippocampus
of mus musculus domesticus

11.45

Nanna Marie Lind:
Linking Personality to Brain Neurotransmission in Animal Models

12.00-12.15

Coffee break

12.15-13.30

AD-models & PET / Chaired by Arne Møller

12.15

Morten Skovgaard Jensen:
Functional changes of synaptic memory in a double transgenic mouse model of Alzheimer’s disease

12.30

Mark J. West:
Structural changes in a double transgenic mouse model of Alzheimer’s disease

12.45

Dirk Bender:
Of Mice and Men: MicroPET imaging of beta amyloid plaque in transgenic mice

13.00

Louise Gyldensted:
MR-studies of AD-patients

13.15

Aage K. Olsen:
The ferret and the mikroPET

13.30-14.00

Lunch

14.00-15.30

RECEPTORS & NEUROTRANSMISSION / Chaired by Paul Cumming

14.00

Uffe Kristiansen:
GABA(A) receptor partial agonists: mechanism of receptor activation

14.15

Jan Sap:
Protein tyrosine phosphatase signaling in the nervous system

14.30

Luciano Minuzzi:
Histamine H3 receptors in the pig brain

14.45

Stig Severinsen:
2,3-Dihydroxybenzoic acid attenuates Kanamycin-induced volume reduction in mouse
utricular type 1 hair cells

15.00

Henrik Hasseldam:
Brain cytokine levels in experimental autoimmune encephalomyelitis (EAE) following treatment
with the cannabinoid receptor agonist WIN 55,212.

15.15

Trine R Larsen:
Protein nitration in organotypic culture models of Parkinson's disease

15.30-15.45

Coffee break

15.45-17.45

CEREBRAL ISCHEMIA / Chaired by Flemming Fryd Johansen

15.45

Christian Hundahl:
Effect of MCAO ischemia on neuroglobin expression in the rat brain

16.00

Jacob Schwartz and Flemming Fryd Johansen:
Vascular receptor upregulation - a novel approach to Stroke pathology

16.15

Rune Skovgaard Rasmussen:
d-Amphetamine promotes cognitive recovery and physical therapy improves fine motor rehabilitation in a rat embolic stroke model

16.30

Flemming Fryd Johansen:
Hypothermia accounts for a significant part of cannabinoid neuroprotection and INFg regulation following cerebral ischemia

16.45

"PET-walking"

17.00

Brent M. Witgen:
Hippocampal quantification after experimentaltraumatic brain injury

17.15

Mette Møller:
Dynamic changes of the corticospinal tract after ischemic stroke detected by MR-fibertracking

17.30

Sys Zoffman:
In vivo studies of the biological activity of functionalised nanoparticles designed for drug delivery usage with focus on delivery to the CNS

17.45

Paul Cumming:
The decline of the Canadian penny

18.30

Hotel check-in

20.00

Dinner
Restaurant L’escale, Åboulevarden 55, 86125315



PROGRAMME
Saturday, June 18th

09.00-10.45

MICROGLIA / Chaired by Bente Finsen

09.00

Lasse Dissing-Olesen:
Axonal lesion-induced reactive microglial proliferation and expression of ICAM-1 in IFN-Beta and vehicle-treated mice

09.15

Reza Khorooshi R:
STAT1 and STAT2 signaling pathway in activated microglia and astrocytes following entorhinal cortex lesion

09.30

Mads D. Pedersen:
Peripheral benzodiazepine receptor expression and PK11195 binding in lesion-induced reactive microgliosis in murine CNS

10.15

Martin Wirenfeldt:
Reactive microgliosis engages distinct responses by microglial subpopulations after minor
CNS injury

10.30

Jesper Kelsen:
Neuroinflammation after transient cerebral ischemia

10.45-11.00

Coffee break

11.00-12.30

NEUROGENESIS / Chaired by Jens Nyengaard

11.00

Torsten M Madsen:
Neurogenesis in the adult rat hipocampus

11.15

Anders Bue Marcussen:
Chronic antidepressant treatment increases hippocampal neurogenesis in rodents

11.30

Thomas Krøigård:
Unbiased estimation of the total number of NeuN positive neurons in the developing neocortex

Jens R. Nyengaard:
FRET-FLIM microscopy

11.45

Jakob Linnet:
High sensation seeking men have increased dopamine release in the right putamen during gambling

12.10

Jette Guldfeldt:
Introducing the new
www.OAKbrain.dk home page

12.25

Arne Møller: Bye-bye




TOP The prefrontal cortex of the Göttingen minipig brain defined by neural
projection criteria and cytoarchitecture

Jacob Jelsing
Research Laboratory for Stereology and Neuroscience,
Copenhagen University Hospital, Bispebjerg, Copenhagen, Denmark


Recently, the debate about the nature and characteristics of the prefrontal cortex (PFC) in non-primate species has resumed. If specific subregions of the PFC are unique to primates, then its role in cognition
and behaviour, and its contribution to disease, can be studied only in these species. Considering the dimensions and large nuclei of the gyrencephalic pig brain, which is comparable to that of humans in gross anatomy, growth and development, we believe pigs may potentially prove useful as an animal model of human frontal lobe function and dysfunction. However, there is to date no available data regarding the localisation of the PFC in the pig brain.
In an attempt to delineate the PFC in the Göttingen minipig brain the distribution of reciprocal thalamocortical projections was investigated using anterograde and retrograde axonal tracing techniques and evaluated in relation to the specific cytoarchitectonic organization. Tracers were visualized using standard immunohistochemistry or evaluated in vivo using manganese (Mn2+) as an MRI paramagnetic tracer. Injections directed towards the mediodorsal thalamus labelled the medial and rostral pole of the frontal lobe as well as anterior cingulate, anterior insular and dorsomedial frontal cortices. Subsequently,
the reciprocity and specificity of these projections was confirmed from injections into the outlined cortices.
Although, the granular layer IV characteristic of primate PFC was not evident our data suggests that the
pig have a structurally divided prefrontal cortex that includes not only features of the medial and orbital areas in primates, but also some features of the primate dorsolateral prefrontal cortex.


TOP Neuron volume in the human neocortex
Anette.K. Stark1, Dorte P. Pelvig1, Henning Pakkenberg1, Morten Møller2 and Bente Pakkenberg1
1 Research Laboratory for Stereology and Neuroscience, Bispebjerg University Hospital, Copenhagen, DK
2 Institute of Anatomy, Panum, University of Copenhagen, DK


The average life expectancy has risen dramatically since the turn of the last century. Lengthening of lifespan has little merit if the quality of life is not preserved, and in the elderly the decline in memory and cognitive abilities is of great concern. With aging we see a small decrease in the total number of neocortical neurons of 9.8% from age 20 to age 90 years, but a gender difference, where men have 16% more neocortical neurons than women.
The aim of this study was to determine the mean volume of neuronal perikaryon and nucleus in human neocortex according to age and gender.
We used a stereological method, the optical rotator, to get an estimation of the three-dimensional size of the neurons in tissue that was isotropically rotated.
The post-mortem material consisted of brains from 19 women average age 63.9 years (18-93 years) and
21 men average age 51.9 years (19-87 years).
We have preliminary results of this study; women have a mean neocortical neuron perikaryon volume of
1364 mm3 and men have a mean neocortical neuron perikaryon volume of 1574 mm3 a significant gender difference of 15% (p=0.02). Women have a mean neocortical neuron nucleus volume of 264 mm3 and men have a mean neocortical neuron nucleus volume of 273 mm3. Women have a decrease in neocortical neuron perikaryon volume by 355 mm3 from the age of 20 to the age of 80 years. Men have a decrease in neocortical neuron perikaryon volume by 331 mm3 from the age of 20 to the age of 80 years. Women have
a decrease in neocortical neuron nuclear volume by 29 mm3 from the age of 20 to the age of 80 years.
Men have a decrease in neocortical neuron nuclear volume by 48 mm3 from the age of 20 to the age of
80 years. None of the age differences were statistically significant. These data are not corrected for in-between gender age and bodysize differences.
In conclusion our preliminary data have shown no difference in neuronal volume decrease with aging and
no gender difference in neuronal nuclear volume, but for perikaryon volume the gender difference shown
in studies of total neocortical neuron number is replicated, men have a 15% larger neocortical perikaryon volume than women.


TOP Neocortical cell number in the common minke whale (Balenoptera acutorostrata) brain
Nina Eriksen & Bente Pakkenberg
Research Laboratory for Stereology and Neuroscience, Bispebjerg Hospital, Bispebjerg Bakke 23,
DK-2400 Copenhagen NV


Cetacean brains are among the least studied mammalian brains. Most research has been carried out on odontocete physiology and anatomi, while the only research on mysticete brains has been done on general morphology. Cetaceans have the largest brain in the Animal Kingdom, but a low Encephalon Quotient (EQ). Encephalisation is a phenomenon that occurred only in the mammalian evolution, where brain size is supposed to increase with increasing body mass. The cetacean brain is very different from the terrestrial mammalian brain in many ways. Like the rest of the whale body, it posses several traits that show adaptation to water. The migration of blowhole from frontal to parietal has changed the shape of the brain and the distribution of the cranial nerves.
This is the first attempt to estimate the neocortical cell number on any species of cetacean - here we use the common minke whale as a model of all mysticetes. Five brains from mature whales were used. Each hemisphere is cut in 2.5 cm slabs using Cavalieri’s method, which is based on unbiased principles for estimating volume of an object. Using a random start the object is cut into parallel sections of equal thickness. The product of the distance between the sections and the total cut area of the same side of
all sampled sections provide an estimate of volume. Neuron and glial numbers are counted using the optical disector, which is a stereological probe for sampling objects according to their number.
A mean number of approximately 14x109 neurons and 10x1010 glial cells were found in neocortex.
This is 2/3 of the human neuron number (19-23x109), but 14 times that of rhesus monkeys (1x109) and
900 times that of mice (1.5x106).


TOP Early induced stress and the consequences on the total neuron number
in the hippocampus of mus musculus domesticus

B.S. Katrine Fabricius, Faculty of Science, August Krogh Institute, University of Copenhagen1,
Research Laboratory for Stereology & Neuroscience2,
Bispebjerg Hospital & Department of Veterinary Pathobiology, laboratory animal science3,
the royal veterinary and agricultural university., 2: Professor dr.med. Bente Pakkenberg 3:
Assistant Professor Thomas C. Krohn.


The aim of the project is to investigate whether experimentally early-induced stress by maternal separation in critical developmental stages in the house mouse, mus musculus, causes behavioural differences and/or neuron cell loss in the mouse hippocampus.
Recently, researchers have found that maternal separation or other pre- or postnatal stress related experiences can change the feeding behaviour, cause high anxiety levels, provoke fear responses and show reduced learning impairments in both the rat and the mouse. Furthermore, a gender difference has been found in both rodent types, where maternal separation causes males to show a higher anxiety level than (diestrous) female.
Two different maternal separation models were used; in the first model the pups were removed from the mother for a minimum of 3 hours per day from postnatal day (PND) 1-14. In the second model the pups
were removed from the mother at PND 9 for 24 hours. In the control litters, the pups went with the dam
at all time undisturbed. The models were performed in both males and females. When the pups reached adulthood, the level of stress was measured with two behavioural tests; an open field test and an elevated plus maze test. The Barnes elevated platform maze were used to test for any damage in the hippocampus.
The maze is equivalent to the Morris water maze, and thus tests for spatial learning and memory.
The mice were sacrificed and the total number, regional volume and density of neurons will be estimated
in the hippocampus using the neuronal optical fractionator design.



TOP Linking Personality to Brain Neurotransmission in Animal Models
Nanna Marie Lind, DVM.
Department of Experimental Medicine, Panum Intitute, University of Copenhagen. nml@cnsr.dk


This talk starts with definition of personality in humans, and addresses the possibility of modelling personality in experimental animals. In particular, the attempt to model the Novelty Seeking (NS) temperament trait (Cloninger et al. 1993) in Göttingen minipigs will be presented.
1) The behavioural response to a novel object was recorded in 12 Göttingen minipigs (test described in Lind et al. 2005a). Subsequently, the same individuals underwent PET scans with the dopamine D2/3 specific radiotracer [11C]raclopride, before and after injection of 1 mg/kg amphetamine. We hypothesised that changes in striatal
[11C]raclopride binding in the amphetamine-challenge paradigm (as described in Lind et al. 2005b) would correlate with the behavioural response to novelty, and that the correlation would be highest in the ventral striatum, a region linked to the rewarding properties of amphetamine and other psychostimulants. The propensity to explore an unfamiliar object (i.e. duration of object contact) was elevated in pigs with high amphetamine-induced dopamine release, primarily in the male pigs.
The results confirm a prior identical study in healthy men (Leyton et al. 2002), thereby supporting the behavioural response of minipigs to a novel object as a possible animal model of the human novelty seeking temperament trait (Lind et al. 2005c).
2) In the same cohort of pigs, learning rate was measured in a Go/No-Go test (test described in Moustgaard et al. 2005). Informal observation of the pigs suggested that fearful animals learned the GNG task faster than less fearful animals. We therefore hypothesised that learning of the GNG task in minipigs could be predicted from their response to novelty, an index of “temperament”. The results showed that pigs with
low behavioral response to novelty learned the GNG task faster than did pigs with a strong behavioural response to novelty, indicated by the tendency to approach novel objects (i.e. number of contacts).
We hypothesise that the critical factor in this relationship is difference in emotional reactivity rather than difference in motivation for exploration (Lind & Moustgaard 2005).
The duration of object contact during the Novel Object test has properties similar to the NS temperament trait in
humans. Future investigations should address whether the number of contacts with a novel object could be an animal homologue of other human temperament traits, such as the Harm Avoidance (HA) trait, and if correlations exists between HA and other neurotransmitter systems.
In summary, The Novel Object Test for Göttingen minipigs provides the means to model the human NS temperament trait. This pig model could prove valuable in future attempts to establish and model behavioural correlates to brain neurotransmission. This would be of particular relevance to research of the pathophysiology of neuropsychiatric disorders.

References:
Cloninger CR et al. (1993). Arch Gen Psychiatry, 50:975-990
Leyton M et al. (2002). Neuropsychopharmacology, 27:1027-1035
Lind NM et al. (2005a). Scand J Lab Anim Sci , in press.
Lind NM et al. (2005b) Brain Res Bull, 65:1-9
Lind NM et al. (2005c) Behavioural Brain Research, accepted
Lind NM & Moustgaard A (2005) Neural Plasticity, accepted
Moustgaard A (2005). Behavioural Processes 2005; 68: 97-102



TOP Functional changes of synaptic memory in a double
transgenic mouse model of Alzheimer's disease

Morten Skovgaard Jensen
The Synapse Project, Institute of Anatomy, University of Aarhus


The â-amyloid hypotheses suggest that an overproduction of â-amyloid and its aggregation in senile plaques is the root cause of Alzheimer’s disease. Neurotoxic effects of â-amyloid and the consequent loss of nerve cells could explain the memory deficits and the cognitive decline that characterize the disease. Newer data indicate that APP processing and the production of â-amyloid is involved in regulation of excitatory synaptic transmission. â-amyloid may therefore interfere with synaptic information processing and memory storage in the brain long before the loss of neurons is significant.
I order to test the latter we investigated synaptic transmission and the induction and the storage of synaptic memory at the age of tree month in normal mice and transgenic mice producing human â-amyloid. The transgenic mice express and produce a mutated form of human APP (APPswe) and the ã-secretase presenilin 1 (PS1) known to course in an early onset of Familiar Alzheimer’s disease.
The production of â-amyloid in the transgenic mice is
elevated from the birth and accumulates over time. The aggregation of â-amyloid into placks occurs at about the 9 month of age.
Synaptic transmission was evaluated by extracellular recording from the CA1 area in the in vitro hippocampus slices preparation. Synaptic potentials were evoked by stimulation of the schaffer-collaterals and population field responses were recorded in the stratum radiatum. Basic synaptic transmission was evaluated by its input-output relationship and was not different when comparing the control mice and the transgenic group of mice.
High frequency stimulation was used to induce synaptic long-term potentiation (LTP) in the synapses.
In normal mice this consist of a transient phase of potentiation which decayed in about half an hour and
a sustained phase lasting more than tree hours. The amplitude of the transient LTP was reduced whereas
the amplitude and saturation level of the sustained form of LTP were not different between the groups.
Post induction test stimulation, using a paired pulse protocol known to destabilize the sustained phase,
was found to be more efficient in reducing the sustained LTP in slices from the transgenic animals.
The transgenic mice show therefore defects in both the induction and the storage of synaptic potentiation month before â-amyloid is aggregating as placks. The data suggest that an overproduction of â-amyloid directly affects the mechanisms underlying potentiation of excitatory synaptic transmission, and consequently may interfere with acquisition and storage of memory.



TOP Structural Changes in Synapses in the Hippocampus of a
Transgenic Model of Alzheimer’s Disease

Mark J. West and Georg Bach Jensen
The Synapse Project, Anatomy, University of Aarhus


We are studying potential changes in the numbers, sizes and types of synapses in the striatum radiatum
of the hippocampal CA1 region of a transgenic mouse model of beta-amyloidosis that produces amyloid plaques that are similar to the type observed in Alzheimer’s Disease (AD). The study is designed to test
the extended amyloid hypothesis of AD, which suggests that one of the initial events, in the cascade of pathological events that leads to AD, is a change in synapses caused by the beta Amyloid protein (Abeta) that is found in abundance in AD brains. We have earlier reported that the stratum radiatum of the CA1 region is particularly vulnerable to AD pathology in humans. We are presently in the process of developing the methodology and equipment required for this analysis. Preliminary data on changes in the number of
CA1 neurons, which will form the background upon which potential changes in synapses are interpreted, indicate that there are no significant differences in the number of CA1 neurons at 12 months of age.
This observation indicates that 12 month old transgenic mice are optimal for our studies in that significant amyloid pathology is present at this time, but there is no sign of the more advanced pathology, i.e. neuron loss change in volume.



TOP Of Mice and Men: MicroPET imaging of beta amyloid plaque in
transgenic mice

Dirk Bender
PET Center, Århus Sygehus

A cardinal pathological characteristic for AD is an increased formation and deposition of plaques in distinguished brain regions. Recently several PET tracers imaging plaques were developed. A new development in PET is scanning of mice and rats in dedicated small sized PET scanners (MicroPET).
It is therefore possible to scan transgenic mice (“AD mice”), which develop plaques like human AD patients. The study will combine the three tools consisting of a pre-clinical animal model, the PET “in vivo autoradiography” and an imaging reagent for AD related plaque to study the suitability of a small animal
PET scanner (MicroPET) for detection of plaques in transgenic “AD mice”, to follow the age dependent formation of these plaques in the transgenetic mice and to evaluate the suitability of a PET tracer for imaging plaque deposition. The outcome of the study will eventually result in valuable information on the potential of this diagnosis approach in human AD patients.
Preliminary results obtained with C-11 labeled PIB in mice are presented.



TOP Perfusion Weighted Magnetic Resonance Imaging in Alzheimer’s
disease and Mild Cognitive Impairment: Preliminary Results

Louise Gyldensted, MD
Neuroradiologic Research Unit, Aarhus University Hospital


Alzheimer’s disease (AD) is associated with several vascular risk factors pointing to a microvascular insufficiency of gray and white matter in AD pathogenesis [1, 2]. Cerebral perfusion measurements in AD with PET and SPECT show hypoperfusion in: Hippocampus, temporo-parietal and frontal cortices [3, 4].
We hypothesize that AD patients have microvascular disturbances of subcortical white matter and that perfusion weighted (PW) MRI with subsequent coregistration can serve as a tool for delineating microvascular perfusion abnormalities across AD patients and thus better characterize disease progression. We studied a group of AD and MCI patients (n=9) and healthy age matched controls (n=18) with contrast bolus PWI MRI. Our initial findings support our hypothesis.
[1] de la Torre,JC: Neurosci.Behav.Rev. 18:397-401, 1994; [2] Brown,WR: Ann.NYAcad.Sci. 903:39-45, 2000; [3] Friedland,RP: JCAT 7:590-98, 1983; [4] Waldemar,G: Cerebrovasc.BrainMetab.Rev. 7:89-130, 1995;


TOP The ferret and the microPET
Aage Kristian Olsen, DVM, Ph.D.
PET-center, Aarhus University Hospital, Noerrebrogade 44, 10c, Dk-8000 Aarhus


We use mainly rodents (mice and rats) in our microPET scanner. However, we like to use the ferret as
a supplement in some brain studies. The weight of the rat brain weighs approximately two grams, and therefore only small amounts of blood can be sampled. The ferret brain weighs 7-10 grams, and the body weight is approximately 1-1½ kg. Therefore, we can get more details when scanning the brain and we can sample more blood in ferrets compared to rats. Furthermore, the cerebral cortex is rough in the ferret brain as in humans. However, there are also some disadvantages in using the ferret as a laboratory animal: Compared to other rodents, ferrets are only rarely used, and therefore much information about ferret
biology is not available. Furthermore, we have some practical problems with the anesthesia of ferrets
and the surgical implantation of catheters. Also the blood glucose seems to vary during the anesthesia.
We are at the moment trying to solve these problems, and furthermore, we are creating a ferret brain atlas. The uptake of 11C-raclopride in the ferret basal ganglia will be shown during the presentation.


TOP GABAA receptor partial agonists: mechanism of receptor activation
Uffe Kristiansen1, Carolina Cannillo1,2, Martin Mortensen1, and Flemming F. Johansen2
1 Dept. of Pharmacology, Danish University of Pharmaceutical Sciences
2 Molecular Neuropathology Group, Institute of Molecular Pathology, University of Copenhagen


The GABAA receptors are ligand gated chloride channels. Activation of the receptors in most cases results
in inhibition of neuronal activity. Partial agonists are defined by their limited ability to activate a receptor (limited efficacy), in this case implying a reduced maximum chloride flux. We have studied activation of GABAA receptors by a number of partial agonist on the single-channel level in order to extract information
on their mechanism of receptor activation. Briefly, the ability to activate the receptor correlates with the ability to stabilize the receptor in the open conformation, while the flux of chloride ions through the open conformation is similar regardless of the efficacy.
Partial agonists compete with full agonists for the receptor binding sites. When a full agonist is displaced
by a partial agonist, the probability of finding the channel open is reduced to a lower level determined by
the partial agonist. In this way, the partial agonist exhibits antagonist properties. It is normally assumed that the potencies of a partial agonist with regard to its agonist and antagonist properties are equal, because both are mediated through binding to the same sites. Our experiments suggest that this is not always the case. Using a generally accepted kinetic model for the receptor together with rate constants extracted from our single-channel experiments, we have simulated the interaction of full and partial agonists and found that the antagonist potency of a partial agonist would be expected to be higher than its agonist potency.
In other words, due to the inherent activation mechanism of the GABAA receptor, the antagonist properties of partial agonists would be effectuated at lower concentrations than the agonist properties.
This may also be true for other ligand gated ion channels with similar activation mechanisms.



TOP Protein tyrosine phosphatase signaling in the nervous system
Jan Sap
Cell regulation Laboratory, Institute of Molecular Pathology, University of Copenhagen

Specific and reversible phosphorylation on tyrosine residues is a major mechanism of intracellular signal transduction. The number of protein tyrosine phosphatases (PTPs) in the genome rivals that of tyrosine kinases, indicating important regulatory roles for this enzyme family. Medically, PTPs are relevant as tumor suppressors and as potential pharmacological targets, yet these possibilities are only beginning to be studied. There is increasing evidence that PTPs play important functions in brain development and synaptic regulation. We will illustrate the possible biological functions of these enzymes based mostly on studies with a ubiquitous PTP, RPTPá. Studies in PC12 cells show that RPTPá can regulate neurite outgrowth in response to NGF, FGF, and EGF in complex ways. Genetic studies in mice reveal unexpected roles in radial neuronal migration, and synaptic plasticity. We will also briefly discuss plans to search for PTPs that regulate neurotrophin sensitivity and neuronal survival


TOP Agonists and Antagonists: do they bind to the same site?
Autoradiographic study of the abundance of agonist/antagonist sites
for histamine H3 and dopamine D2/3 receptors.

Luciano Minuzzi
PET Center, Århus Sygehus

Introduction: G-protein coupled receptors are a large family of receptors that mediate transmembrane signal transduction in response to the binding of many neurotransmitters, peptides, hormones and autacoids. Agonist binding changes the G-protein complex, increasing the activity of enzymes which in turn regulate second messengers. When there is no dissociation of the G-protein complex, agonists bind with high affinity to the receptor. Upon agonist binding, the G-protein is activated and the receptor converts to a low affinity state for agonists. Antagonist binding is unaffected by G-proteins. Since only the agonist fraction is functional, endogenous neurotransmitter and drug efficacies are determined by agonist potency on the receptors in the high affinity state.
On the basis of various studies in vitro and in vivo, the fraction of dopamine receptors in the high affinity state has been estimated to be 40%. However the function of the receptors in the low affinity state is uncertain. In order to obtain a better understanding of dopamine D2/3 agonist binding, we carried a series
of experiments to test the sensitivity of [3H]NPA (D2 agonist) and [3H]raclopride (D2/3 antagonist) in rat brain cryostat section to LSD competition, and their saturation binding parameters. In another study, we used quantitative autoradiography to measure the saturation binding parameters for [3H]N-M-HA (H3 agonist) and [125]IPP (H3 antagonist) in several regions of cryostat sections from brain of Landrace pigs.
Methods: Twenty m m-thick cryostat sections from rats (Lewis/Mol strain) and four adult female Landrace-Yorkshire pigs were used in the experiments. Rat brain sections were incubated with 1 nM [3H]NPA or 2 nM [3H]raclopride along with LSD at final concentrations ranging from 10-13 M to 10-4 M. Addition of 100µM guanylyl-5'-imidodiphosphate (Gpp(NH)p) induced dissociation of the G-protein complex changing the dopamine receptor to a state with low affinity for agonists. To assess comparable processes in the case
of histamine H3 receptors, saturation binding experiments were carried out in pig brain sections incubated with [3H]N-M-HA or [125]IPP. One-site and two-site models were fitted to the displacement series and
the saturation binding experiments for the calculation of the IC50s, Bmax and Kds (Sigma Plot 8.02).
Results and Discussion: Preliminary results will be presented and discussed in the context of PET competition models
.


TOP 2,3-Dihydroxybenzoic Acid Attenuates Kanamycin-induced Volume
Reduction in Mouse Utricular Type I Hair Cells

Stig Å. Severinsen1, Mette Kirkegaard2, Jens R. Nyengaard1
1 Stereology and Electron Microscopy Research Laboratory, Institute of Clinical Medicine, University of Aarhus, Denmark
2 Center for Hearing and Communication Research, Karolinska University Hospital, Stockholm, Sweden


Sensory hair cells are delicate structures which can be damaged by exposure to aminoglycosides.
The aim of this study was to estimate cellular quantitative changes in the utricular balance organ of mice
to assess a possible damage to cells after treatment with the aminoglycoside kanamycin. Antioxidant therapy with 2,3-dihydroxybenzoic acid (DHB) was also introduced to attenuate the cell damaging effect
of kanamycin.

Mice were injected twice daily with either saline, kanamycin or kanamycin + DHB for 15 days and perfusion fixed three weeks after last injection. Total volume of the utricle as well as number of hair and supporting cells was estimated using stereological methods. Volume of hair cells (HCI & HCII), supporting cells (SC)
and neural elements were estimated on electron micrographs.
Mean volume of the utricle was 3.65 · 10-3 mm3 (0.07) in control animals and 3.50 · 10-3 mm3 (0.06) in kanamycin + DHB-treated animals. In animals treated with kanamycin the volume was reduced to 3.14 ·
10-3 mm3 (0.04) which was significantly different from the two other groups.
Although hair and supporting cell numbers remained unchanged regardless of treatment, cell volume was significantly affected. Mean volume of HCI was 270 microm3 in control animals. Kanamycin-treated animals had a HCI mean volume of 209 microm3 and were significantly different from kanamycin + DHB-treated animals (P=0.04), which had a HCI mean volume of 286 microm3, but only tended to be different from controls (0.09). Mean volume of HCII and SC did not differ significantly between the groups (P0.05).
We did not find any apoptotic cells (no caspase-3 reactivity).
This experiment demonstrates that two kanamycin-injections of 900 mg/kg/day do not alter the number
of sensory hair cells in the utricular macula of mice. However, a significant decrease in volume of the utricular sensory epithelia indicates that the tissue was affected by the kanamycin treatment.
Mean volume of HCI and total volume of the utricular macula did not decrease in animals co-treated with
the antioxidant DHB, indicating that antioxidant therapy could be a successful way of otoprotection against aminoglycoside-induced inner ear damage.


TOP EAE, Cannabinoids & Cytokines
Henrik Hasseldam
Molecular Neuropathology Group, University of Copenhagen, Copenhagen, Denmark


Molecular Neuropathology Group, Institute of Molecular Pathology, University of Copenhagen
Cannabinoids are increasingly in focus as a possible symptomatic treatment for Multiple Sclerosis (MS). MS patients describe a relief of pain, tremor and paralysis when smoking marihuana. These effects are supported by clinical studies showing minor overall improvements in the general well-being of MS patients.
With this in mind we have established an animal model, Experimental Autoimmune Encephalomyelitis (EAE), which shares substantial clinical and pathological characteristics with MS. In order to explore the effects
of symptomatic cannabinoid treatment on the development and severity of EAE, we set up a treatment regimen which included daily i.p. injections (2.5 & 5.0 mg/kg/24h) with the synthetic cannabinoid analogue WIN-55,212-2, initiated at symptom debut.
The results clearly demonstrated an effect on the neuropathological level, with regards to a reduction in
the amount of inflammatory cells and degree of demyelination. This was especially true for the high WIN-55,212-2 concentration. Furthermore, we wanted to test whether the cannabinoid treatment, had an influence on the concentration of cytokines in the CNS. We focused on the pro-inflammatory cytokines TNF-á and IFN-ã, and actually observed a significant increase following cannabinoid treatment. This is somewhat surprising in the sense that both cytokines have been shown to be toxic to neurones and oligodendrocytes, and to augment the inflammatory activity in the CNS. On the other hand, the presence of these cytokines at later time points has been shown to induce programmed cell death in T-cells and promote remyelination, thus reducing the disease burden in animal models of MS.



TOP Protein nitration in organotypic culture models of Parkinson's disease
Trine R. Larsen1,2, Ann-Sofi Peterson3, Kenneth Caidahl3, Peter Roepstorff2, Jan Bert Gramsbergen1.
1 Anatomy and Neurobiology, Institute of Medical Biology, University of Southern Denmark.
2 Biochemistry and Molecular Biology, Faculty of Science and Engineering, University of Southern Denmark.

3 Clinical Physiology, Sahlgrenska University Hospital, University of Göteborg, Sweden.

Objectives
Nitrated proteins have been detected in nigral Lewy bodies of Parkinson’s disease (PD) patients, but it is unclear whether protein nitration is a critical event in the degeneration of dopaminergic neurons. Here we quantified protein-bound 3-nitrotyrosine (3-NT) in toxin-treated organotypic, mouse ventral mesencephalic (VM) cultures and correlated this with dose-dependent dopamine depletions.
Materials and Methods Organotypic VM cultures of embryonic day 12 mice (CBL57/bl6) were grown for 3 weeks and then treated (acute: 24 or 48 hours, chronic: 3 weeks) with the peroxynitrite donor 3-morpholino sydnonimine (SIN-1), 1-methyl-4-phenylpyridinium (MPP+) or rotenone, or co-treated with MPP+ and the nitric oxide synthase inhibitor N-nitro L-arginine methyl ester (L-NAME). Protein-bound 3-NT was quantified using a novel gas chromatograpy/negative chemical ionisation tandem mass spectrometry technique.
Tissue dopamine and medium 3,4-dihydroxyphenylacetic acid (DOPAC) levels were assessed by HPLC with electrochemical detection.
Results Acute SIN-1 or MPP+ treatments caused dose-dependent protein nitration reaching a maximum
of 8-fold by 10 mM SIN-1 or 2-fold by 10 µM MPP+. Chronic MPP+ or rotenone treatments caused maximum protein nitration by 1 µM (2-fold) or 50 nM (4-fold) respectively. Co-treatment with L-NAME (300 µM) prevented protein nitration by acute MPP+.
Conclusions Protein nitration and dopamine depletion by MPP+ or rotenone treatments are closely related, but inhibition of protein nitration did not prevent dopamine depletion in the acute MPP+ model. Whether protein nitration plays a role in dopamine depletion and neuronal cell loss under chronic conditions remains
to be investigated.



TOP Does neuroglobin protect neurons after transient cerebral ischemia?
C. Hundahl1+; J. Kelsen2+; L.C.B. Rønn3; and J.R. Nyengaard4
1 Department of Zoophysiology, Institute of Biology; 2Water and Salt Research Centre; 4Stereology Research Lab, University of Aarhus; and 3NeuroSearch A/S, DK-2750 Ballerup, Denmark

+These authors contributed equally to this work.

Introduction: Brain ischemia due to stroke is a major cause of brain injury leading to disability and death. Neuroglobin (Ngb) is a novel characterized heme globin primarily expressed in retinal nerve cells and at very low levels in endocrine active brain regions in vertebrates. When artificially over-expressed, Ngb can reduce the infarct size in a transient model of Middle Cerebral Artery occlusion (MCAo) in rats. Hence modulation
of Ngb expression may have a significant potential in new treatment strategies of stroke. However, it is not known whether a protective effect is present at physiological levels of Ngb.
Materials and methods: Thirteen Spontaneously Hypertensive Rats (SHRs) subjected to either ninety minutes of transient MCAo or sham surgery on the right side were euthanized on day eight after surgery.
We used free-floating immunohistochemistry with polyclonal and monoclonal antibodies directed against
Ngb and a neuronal marker (NeuN), respectively. Design-based stereologic quantification of Ngb and NeuN positive cells in the striatum of all animals was performed using the optical fractionator.
Results: The ischemic damage affected primarily striatal structures and constituted 16.6 mm3 in the MCAo rats and was not present in the sham rats (p<0.005) . We a significant lower number of Ngb positive neurons in MCAo (n=7) rats compared to sham (n=6) ( p>0.005). These findings suggest that Ngb does not have a protective effect at physiological levels. Furthermore, Ngb expression is mainly confined to the hypothalamus and amygdale, which is not directly affected by the ischemic lesion. The level of expression was also lower in the ischemic hemisphere when compared to the non-ischemic hemisphere of MCAo rat brains.

Conclusion: Ngb, expressed at physiological levels after transient MCAo in SHRs, does not provide protection against ischemic injury.
Support by: EU (grant QLG3-CT-2002-01548). No conflict of interests.


TOP Temporary cerebral ischaemia upregulates the 5-HT(1) receptor
in the middle cerebral artery

Jacob Hansen-Schwartz1,2, Flemming Fryd Johansen2, Lars Edvinsson1,3
1 Department of Experimental Research, Glostrup University Hospital, Glostrup, Denmark
2 Institute of Molecular Pathology, University of Copenhagen, Copenhagen, Denmark
3 Department of Internal Medicine, University of Lund, Lund, Sweden


Stroke gives rise to an immediately infarcted area surrounded by an area of critically perfused neural tissue ('area at risk'); the fate of this tissue being dependent on increased perfusion subacutely.
Using experimental temporary occlusion of the middle cerebral artery (MCA) in the rat we studied the possible upregulation of the 5-HT(1) receptor in the MCA. Experimental stroke: The MCA of an anaesthetised rat was exposed and temporarily occluded with a hook for 120 mins. Afterwards the rat was revitalised.
In vitro pharmacological examination: After two days the rat was killed and the MCA's were harvested and suspended on wires for measurement of contractile properties. Selective 5-HT(1) agonists and antagonists were used to study contractile responses. Contractile responses to 5-HT(1) stimulation were clearly enhanced after stroke (compared to the contralateral MCA). This receptor upregulation implies an increased sensitivity towards the endogenous agonist 5-hydroxytryptamine. It has earlier been shown that temporary occlusion leads to upregulation of a contractile ET(B) receptor. The combined upregulation of contractile receptors may further reduce the blood supply to the area at risk, thus, increasing the infarct size with subsequent increased neurological disability.


TOP D-Amphetamine promotes cognitive recovery and physical therapy
improves fine motor rehabilitation in a rat embolic stroke model

Rune Skovgaard Rasmussen, MA; Karsten Overgaard, MD; Elisabeth S. Hildebrandt-Eriksen, PhD; Gudrun Boysen, MD, DMSc.
Neurovascular Research Laboratory, University Hospital of Copenhagen, Teilum Building

Background and Purpose: The purpose of this study was to examine effects of d-amphetamine and physical therapy alone or combined in terms of fine motor performance, gross motor performance and cognition after middle cerebral artery thromboembolization in rats.
Methods: Seventy-four rats underwent surgery and 59 were embolized in the right carotid territory with
an embolus and randomly assigned to: 1) SHAM (non-embolized, saline), 2) CONTROLS (embolized, saline), 3) D-AMPH (embolized, d-amphetamine), 4) THERAPY (embolized, saline + physical therapy) and 5) D-
AMPH+THERAPY (embolized, d-amphetamine + physical therapy). Groups 3-5 received d-amphetamine treatment and/or physical therapy on days 1, 3, 5 and 7 after surgery. Animals from all groups were re-tested during days 21 to 28 after surgery.
Results: No differences in infarct volumes were observed between groups of embolized animals. When evaluating performances on days 21 to 28 after surgery, SHAM and THERAPY had better fine motor performance than CONTROLS (P < 0.05), while SHAM and D-AMPH achieved better cognitive performance than CONTROLS (P < 0.05). No significant differences were observed between any groups regarding gross motor performance.
Conclusions: After embolization physical therapy improved fine motor performance and d-amphetamine accelerated rehabilitation of cognitive performance.



TOP Hypothermia accounts for a significant part of the neuroprotection
provided by cannabinoids following cerebral ischemia.

Peter K. Bonfils, Jakob Reith, Henrik Hasseldam, and Flemming Fryd Johansen*
Molecular Neuropathology Group, University of Copenhagen, Copenhagen, Denmark


Cannabinoids have neuroprotective potentials, and the expression of endocannabinoids as well as cannabinoid receptors are induced after cerebral ischemia. They also induce hypothermia by lowering the hypothalamic set point. We have investigated the significance of such hypothermia in ischemic neuroprotection following systemic administration of WIN 55,212-2, a synthetic cannabinoid receptor agonist. Results showed that WIN 55,212-2 significantly reduced infarct volumes of rats subjected to focal cerebral ischemia (middle cerebral artery occlusion) and significantly decreased ischemic CA1 damage in rats subjected to global cerebral ischemia (two-vessel occlusion). A significant (approximately 50%) part of this neuroprotection was provided by WIN 55,212-2 induced hypothermia (33.7 1.1C / 34.9 1.6C), because prevention of hypothermia by maintaining body core temperatures between 37.0-38.0C dissolved the neuroprotective effect into a hypothermic component and an unidentified component. Finally, the ability of WIN 55,212-2 to reduce levels of the proinflammatory cytokine IFN in the infarcted hemispheres of rats subjected to focal cerebral ischemia required hypothermia.
We conclude that cannabinoids are reliable candidates for drug induced hypothermia and neuroprotection. These neuroprotective effects could provide the basis for potential therapeutic uses of cannabinoids and/or endocannabinoids in stroke.



TOP GFP-transgenic mice to quantify hippocampal Inhibitory Interneuron
Loss by stereology after fluid percussion Brain Injury.

B. M. Witgen1,2, J. Lifshitz3, J. R. Nyengaard1, M. S. Grady2.
1 Stereology and Electron Microscopy Research Laboratory, Aarhus Denmark;
2 Department of Neurosurgery, University of Pennsylvania, Philadelphia, PA;
3 Department of Anatomy and Neurobiology, Virginia Commonwealth University, Richmond,VA.


Susceptibility of hippocampal neurons to human brain injury can also be identified in experimental models. After lateral fluid percussion brain injury in the mouse, design-based stereology confirmed a uniform loss of 25-35% of all neurons in the four major subregions by one week post-injury, which does not progress by
one month. Since excitatory and inhibitory networks combine to establish hippocampal function, the neuronal loss could be all excitatory neurons, all inhibitory neurons, or a combination of the two populations.
To begin to address the nature of hippocampal neuronal loss after TBI, we have taken advantage of GFP-GAD ( FVB-TgN(GadGFP)45704Swn) transgenic mice to quantify the remaining population of somatostatin-positive inhibitory interneurons in the hippocampus using combined transgenic-fluorescent-stereology.
At one week, the brains of brain-injured and uninjured control mice were processed for stereological quantification of GFP-positive somatostatin-positive inhibitory interneurons in the hilus. Uninjured control mice had 1140 (CV=0.06) somatostatin-positive interneurons, whereas brain-injured mice 900 (CV=0.05).
In the hilus at one week after injury, 21% of the interneurons are lost, but previous data shows a 34% total neuronal loss. Consequently, the proportion of somatostatin-positive inhibitory interneurons in the hilus increases after brain injury (9.9% to 11.9%), with potential functional implications. Further studies address the remaining hippocampal subregions and other inhibitory interneuron subpopulations.



TOP Dynamic changes of the corticospinal tract after ischemic stroke
detected by MR-fibertracking

Mette Møller1,2, Jesper Frandsen1, Grethe Andersen3, Dora Zeidler1, Albert Gjedde1,2,
Peter Vestergaard-Poulsen
1 Center of Functionally Integrative Neuroscience1, Aarhus University, PET-Center, Aarhus University Hospital
2 Department of Neurology3, Aarhus University Hospital, Denmark


Introduction
The integrity and connectivity of nerve fiber tracts in the brain are important in assessing plastic changes related to
functional recovery and to obtain prognostic information and formulate future therapeutic strategies for stroke patients.
Previous imaging studies have shown that the adult brain after ischemia can regenerate and compensate for motor deficits by plastic changes, though demonstration of wallerian degeneration is associated with more permanent neurological deficts.
To our knowledge, the integrity of the corticospinal tract in a longitudinal study of stroke from the onset of the acute stroke and throughout rehabilitation has never previously been documented in humans.
Using diffusion measurements (DTI) and computer based 3D axonal fiber tracking algorithms in correlation with neurological motor scale we hypothesized that changes in axonal integrity along the corticospinal tract after stroke can be detected as reduction in fractional anisotropy (FA-index) and that a sustained low FA-index is indicative of axonal loss and correlates with poor motor outcome. Finally we speculated whether a reduction of FA-index is associated with a low density ratio (ipsi/contra-lesional) of the tracked corticospinal fibers.
Methods
Five right-handed patients with first-time subcortical ischemic infarcts and motor deficits were tested with Medical Research Council (MRC) and MR-scanned on day 1-4, 30 and 90 post-stroke. Serial DTI was performed using a birdcage head-coil and double spin echo single shot EPI at 1.5 T, employing 17 isotropically-distributed directions, and a b-factor of 1000 s/mm2,
with additional b-factor=0 s/mm2 images. Maximum gradient strength was 36 mT/m. 50 slices of 3.3 mm thickness were acquired, covering a 24 cm FOV in a 128x128 matrix. TR/TE =17000/84 ms. The sequence was repeated four times for a total 22 min acquisition time. The eigensystem was calculated from the diffusion tensor in each voxel using diagonalization. Fiber tracking was calculated with the FACT algorithm.
Results
The temporal evolution of the ratio (ipsi/contralesional) of FA-index was unchanged (above 0.9) in the four patients with good outcome (MRC=4), whereas a decline was seen in the patient with poor outcome (MRC=1.2) The reduction of the FA-index was associated with a decreased intensity of the affected cerebral peduncle in the FA-maps and a low density ratio of the tracked fibers indicative of axonal loss.
Discussion
The novel findings seem to indicate an association between motor function and reduction in both FA-index and density of the tracked fibers and that these parameters appear to be sensitive of structural changes in the corticospinal tract after stroke.
The data are preliminary based on five patients and inclusion of more patients and a methological study on the connection between FA-index and the fiber-tracking algorithm is planned.



TOP In vivo studies of the biological activity of functionalised nanoparticles
designed for drug delivery usage with focus on delivery to the CNS.

Sys Zoffman
Stereology and Electron Microscopy Research Laboratory, Aarhus Denmark

Development and usage of nano-scale particles as carriers of drugs have attracted considerable interest
as potential diagnostic and therapeutic agents.
Positively charged polymeric molecules such as chitosan are able to encapsulate negatively charged nucleic acid molecules. Furthermore, the core can be encapsulated by a second type of polymer, which increases the bloodstream circulation and potentially also the transfection activity. Incorporation of small interfering RNAs (siRNA) into polymer-based nanoparticles constitute a possible solution as a drug for treating neurodegenerative disorders (Alzheimer’s disease and Pakinson’s diseases).
However, the blood-brain barrier (BBB) constitute a major obstacle in the delivery of drugs to the central nervous system (CNS) as only small, lipid-soluble molecules are allowed to pass the BBB.
It is therefore of great interest to develop particles of nano-scale size, which can either diffuse freely through the BBB or which are functionalised with ligands to be transported with receptors present in the BBB. In this study we have used an EGFP (Enhanced Green Fluorescent Protein) expressing mouse model
to test the delivery and activity of nasally administered chitosan-encapsulated siRNA against the EGFP
mRNA to the mouse olfactory bulb and brain. We are still facing technical problems and would like to know more about ligands which are suitable candidates for crossing the BBB.



TOP The decline of the Canadian penny
Paul Cumming
Centre for Functionally Integrative Neuroscience, Aarhus

Introduction: Kinetics can mean the study of the effects of forces on material objects, but in the context of chemistry and biochemistry often refers to the laws governing rate of change in concentration of a molecule. The mathematics underlying simple kinetic analysis is simple indeed; One calculates the rate of change in the concentration of a chemical product, or the rate of entry of a tracer into a metabolic compartment as a function of the concentration of precursor and a first order rate constant. While a biochemist can often keep the concentration of a precursor constant in the course of the experiment, this
is not the case in PET studies; An intravenous bolus of tracer results in a peak concentration occurring one minute after injection, followed by a decline, which can be modeled as a series of parallel first order processes, i.e. mixing in the blood, distribution in body tissues, and metabolism or renal elimination.Plasma pharmacokinetics is a well-established field for describing the fate of a PET tracer or indeed any medication. The same approach can be used for the study of diverse other systems, in which the concentration or abundance of something (minke whales, coins in circulation) changes as a function of time, according to some orderly law. Historians have used this approach to attempt to reconstruct ancient economics, on the basis of large sample of coins, collected as "hoards". Surprising, this can also be done at home, and without a metal detector.
Methods: A sample of 1600 Canadian pennies was hoarded in a large pickle jar during a period of two years. The sample was stratified by age, and corrected for the annual output of pennies from the Royal Canadian Mint. Population survival curves were calculated for the sample. In another study, a hoard of 400 American coins in circulation in Canada was likewise examined.
Results: The survival curve of the Canadian penny revealed two phases; an initial rapid phase, reflecting the intrinsic half-life of the coin (five years). Some 40% of the coins disappeared with a much slower half-life, close to 20 years. This may reveal the re-entry of hoarded coins into circulation after a delay of two decade. The total hoard is calculated to consist of 17,000,000,000 coins. The American penny survival curve revealed an early growth function (Tau), indicating the delay for entry into circulation. The population then declined with a half-life of 20 years, suggesting that surviving pennies enter into the pool with slow turnover, i.e. pickle jars.


TOP Axonal lesion-induced reactive microglial proliferation and expression
of ICAM-1 in IFN-Beta and vehicle-treated mice

Dissing-Olesen L., Dalmau I., Ladeby R., Nielsen H. H., Finsen B.
Medical Biotechnology Center, University of Southern Denmark,
Winsløwparken 25, DK-5000 Odense C, Denmark


Demyelination and axonal degeneration are prominent in multiple sclerosis (MS). Interferon (IFN)- is known
to have a beneficial therapeutic effect with relapsing remitting MS patients and is known to reduce microglial proliferation in vitro and endothelial expression of the intercellular adhesion molecule (ICAM)-1 in vivo in rodents.
A murine model for axonal degeneration was used to investigate if IFN- reduces the axonal-lesion induced microglial reaction, which may contribute to disease progression. Transection of the entorhino-dentate perforant path-projection results in an anterograde axonal (Wallerian) and terminal degeneration that induces a region-specific activation and proliferation of microglia in the dentate gyrus. By applying double-label immunohistochemistry for the macrophage antigen (Mac)-1 and the proliferation marker bromodeoxyuridine, injected one hour prior to euthanasia, we found that 25% of all lesion-reactive microglia were proliferating 3 days post-lesion, at which time the microglial cell population had increased 3-fold in lesioned mice compared to controls. Interestingly, at this time 50% of all the lesion-reactive microglia expressed the co-stimulatory molecule the ICAM-1. Fluorescence-double labeling immunohistochemistry for Mac-1 and ICAM-1 demonstrated co-localisation.
Treatment with human (h)IFN-beta (Rebif) had no effect on the microglial morphology and no statistically significant effect on the total number of reactive microglia, the number of actively proliferating microglia, or the ones coexpressing ICAM-1 (IFN-treated, n = 7; vehicle-treated, n = 7, P 0,05 for all comparisons). As the absence of effect might be explained by lack of penetration of IFN- across the blood brain barrier or lack of effect of hIFN- on murine cells, a conclusion about the effect of IFN- on axonal lesion-induced microglial activation can therefore not yet be drawn.



TOP STAT1 and STAT2 signaling pathway in activated microglia and
astrocytes following  entorhinal cortex lesion

Khorooshi R, Owens T.
Medical Biotechnology Centre, University of Southern Denmark, Odense, Denmark


Microglia and astrocytes in the outer molecular layer (OML) of the hippocampal dentate gyrus are activated in response to entorhinal cortex lesion (ECL). Signals for glial response are not well defined. Several cytokines that may trigger these responses signal through receptor associated signal transducer and activator of transcription (STAT). A role for type 1 interferon has been proposed. Type 1 interferon act via a receptor that is associated with STAT1 and STAT2 signaling pathway. The present study was therefore designed to investigate whether ECL induces activation of STAT1 and STAT2 in OML. The preliminary results showed induction of STAT1 in reactive microglia and STAT2 in astrocytes within the denervated hippocampus 3 days after ECL. These findings indicate the involvement of type 1 interferon specific signaling pathways (STAT1 and STAT2) in lesion-induced glial activities. In future studies we will ask whether STAT signaling pathways play a role in the initiation of immune responses to axonal injury at earlier time, and in different mouse models.


TOP Peripheral benzodiazepine receptor expression and PK11195 binding
in lesion-induced reactive microgliosis in murine CNS

Mads D. Pedersena, Luciano Minuzzib, Martin Wirenfeldt 1, Michael Meldgaard 1, Paul Cumming 2 and Bente Finsen 1
1 Medical Biotechnology Center, University of Southern Denmark, Odense C, Denmark, and
2 Aarhus University PET Centre, and Center for Functionally Integrative Neuroscience, Aarhus University Hospital, Aarhus, Denmark


The peripheral benzodiazepine receptor (PBR) binds the ligand PK11195 with high affinity.
The receptor, which is located primarily to the outer mitochondrial membrane, is composed of three subunits: the isoquinoline-binding protein (18 kDa), the voltage dependent anion channel (32 kDa), and the adenine nucleotide transporter (30 kDa). The receptor has roles in steroid production, energy metabolism, cell survival and growth. A large number of studies have reported an increase in PK11195 binding following damage to the CNS. This increase in binding has been attributed to an increase in expression of the PBR by activated microglia and infiltrating macrophages.
Adult C57BL/6 mice were subjected to a stereotactic transection of the entorhinal-hippocampal perforant path (PP) projection resulting in a highly characteristic microglial reaction in the PP-terminal zones in the dentate gyrus and the hippocampus proper. PBR binding was analysed in brain sections and PBR mRNA expression in hippocampal homogenates obtained from mice with 2, 5 and 10 days survival postlesion and sham-operated and unoperated controls.
For the PBR ligand PK11195, Bmax and Kd were established in the ipsi- and contralateral dentate gyrus,
the ipsilateral CA3 and CA1, and in the cortex, caudate nucleus, dorsolateral thalamus, superior colliculus, inferior colliculus, fimbria, and cerebellum. Bmax displayed a 3-fold increase 5 days post lesion in the dentate gyrus, which correlates with the time of maximal activation of Mac-1 immunoreactive microglia. Quantitative rtPCR revealed peak expression of PBR mRNA 5 days post lesioning, corresponding to maximal expression of Mac-1 mRNA. In addition, rtPCR analysis using exon-specific primers, indicated the presence of two splice forms, a long form consisting of all 4 exons, and 3-fold more abundant short form consisting of exon 2 and 3. Comparison of Bmax in different brain regions revealed an up to 3-fold difference between regions, the fimbria showing the strongest and the inferior colliculi the smallest binding affinity.
These preliminary data are presently being supported by inclusion of larger numbers of mice in the experiment and inclusion of information on the cell-specific expression of PBR.



TOP Reactive microgliosis engages distinct responses by microglial
subpopulations after minor CNS injury

Martin Wirenfeldt1, Alicia Anne Babcock2, Rune Ladeby1, Kate Lykke Lambertsen1, Frederik Dagnaes-Hansen3, Robert Graham Quinton Leslie4, Trevor Owens1,2 and Bente Finsen1
1 Medical Biotechnology Center, University of Southern Denmark, Winsløwparken 25, DK-5000 Odense C, Denmark
2 Neuroimmunology Unit, Montreal Neurological Institute, Montreal, Quebec, Canada H3A 2B4
3 Department of Medical Microbiology and Immunology, University of Aarhus, Wilhelm Meyers Allé 240, DK-8000 Aarhus C, Denmark
4 Immunology and Microbiology, Institute of Medical Biology, University of Southern Denmark, Winsløwparken 21, DK-5000 Odense C, Denmark


Microglia are bone marrow-derived cells that constitute a facultative macrophage population when activated by trauma or pathology in the CNS. Endogenous CNS-resident microglia as well as exogenous (immigrant) bone marrow-derived cells contribute to reactive microgliosis. This phenomenon raises fundamental questions about the cellular composition, kinetics and functional characteristics of the reactive microglial cell population in the CNS. Bone marrow chimeric mice reconstituted with green fluorescent protein expressing (GFP+) donor bone marrow cells were subjected to a selective axonal degeneration resulting in a localized microglial reaction in the hippocampus. Flow cytometric evaluation of individual microdissected hippocampi demonstrated small, but consistent, increases in the proportion of immigrant GFP+ microglia (CD11b+CD45dim) by 3 and 5 days post-lesion. Seven days post-lesion, however, approximately 13% of microglia in lesion-reactive hippocampi were bone marrow-derived. Immigrant microglia expressed lower levels of CD11b than resident microglia in bone marrow chimeric mice, forming a distinct subpopulation on CD11b/CD45 profiles. In addition a subpopulation of resting and activated CD11b+ microglia, primarily of resident origin, expressed the haematopoietic stem cell marker CD34. Our results show that distinct subpopulations of microglia respond to minor CNS injury, and suggest that this heterogeneity in microglial response encloses functional consequences for repair and possibly therapy.


TOP Neuroinflammation after transient cerebral ischemia
Jesper Kelsen, MD1, 2
1The Water and Salt Research Centre, University of Aarhus, DK-8000 Aarhus, Denmark
2 Clinical Institute, University Hospital of Aarhus, DK-8200 Aarhus N, Denmark


There has been a static view upon the inability of human adult brain tissue to renew itself. However, the discovery of neurogenesis in the adult human hippocampus has led to considerable research in the potential to regulate human neurogenesis. Both the hippocampal dentate gyrus Granule Cell Layer (GCL) and the Subventricular Zone (SVZ) house neural stem cells with the potential of differentiating into glia or neuronal cells. Incorporation of the thymidine analog, 5-bromo-2´-deoxy-uridine (BrdU) is the classical method used to prove the proliferation of neural stem cells in adult brain tissue. Recently, infiltration with endogenous precursor cells in an infarcted area, has been documented in an adult rat model of transient Middle Cerebral Artery occlusion (tMCAo). The proces of neurogenesis is stimulated by brain damage like degeneration, inflammation and ischemia.
The innate neuroinflammatory response to brain injury delivered by activated microglia is considered as a doubleedged sword. A complex interplay between astrocyte glutamate release and activated microglia is proposed to cause neurotoxicity. Recently, the deleterious effects of microglial secretion of the proinflammatory mediator, IL-6 have been adressed in regard to hippocampal neurogenesis. Blockage of neuronal inflammation with indomethacin or microglial activation with minocycline has
effectively restored hippocampal neurogenesis in rats subjected to lipopolysaccharide (LPS) induced systemic inflammatory respons syndrome (SIRS) or cranial irradiation.
In this PhD study neuroinflammation and neurogenesis after tMCAo is being investigated in two different rat strains. Unbiased stereological methods are used for the immunohistochemical quantification of hippocampal BrdU incorporation and an activated microglia marker (ED-1). Further the possible beneficial effects of selective COX-2 inhibition after tMCAo is evaluated with immunohistochemistry, quantitative RT-PCR and MRI.



TOP Neurogenesis in the adult rat hipocampus
Torsten M. Madsen, M.D., Ph.D.
Center for Basic Psychiatric Research, Aarhus University Hospital Stereology and Electron Microscopy Res. Lab., Aarhus University


Psychiatric treatment and neural plasticity.

Hippocampal neurogenesis is increased after administration of antidepressant drugs as well as seizures, indicating a dynamic regulation of this process. To further investigate this important phenomenon, studies are underway to quantify changes in the number of synapses in discrete regions of the rat brain after antidepressant treatment.
Also, the molecular underpinnings of the neural plasticity are investigated:
After electroconvulsive seizures, b-catenin, an important component of the Wnt pathway, is increased in the hippocampal dentate gyrus, in places where cell proliferation also occurs. Given that electroconvulsive seizures are commonly used for the treatment of intractable depression, b-catenin and the Wnt pathway may be potential therapeutic targets for psychiatric disorders.



TOP Chronic antidepressant treatment increases hippocampal
neurogenesis in rodents

Anders B. Marcussen1,2, Peter Flagstad2, Flemming F. Johansen1, Paul E.G Kristjansen1 and Ulrica Englund2
1 Institute of Molecular Pathology, University of Copenhagen, Denmark
2 H. Lundbeck A/S, Pharmacology Target Research, Copenhagen, Denmark


Recently, it has been hypothesized that generation of new nerve cells (neurogenesis) in the hippocampus is necessary for the effect of antidepressant treatment. This hypothesis is based on findings from pre-clinical studies, showing that several modalities of chronic antidepressant treatment increase hippocampal neurogenesis (e.g. Malberg et al., 2000).
In the current study, we treated mice and rats with fluoxetine (10 mg/kg) or vehicle for 28 days prior to being tested in the NSF assay. Proliferating cells were detected using the thymidine analogue BrdU, which becomes incorporated into the DNA of dividing cells. The level of neurogenesis was analysed at day 28 using immunohistochemical techniques and microscopical analysis.
The behavioural effect of chronic as well as acute antidepressant treatment was examined using the NSF test. This anxiety-related behavioural test is able to detect an effect of chronic, but not acute, antidepressant treatment in rats and mice (Bodnoff et al. 1989; Santarelli et al. 2003).
The results showed that fluoxetine-treatment had a significant neurogenic effect in mice. In rats, a tendency towards an increase in neurogenesis was observed after the fluoxetine treatment, although this did not reach statistical significance. The chronic drug-treatment resulted in a significant behavioral effect using the NSF test in rats, but not in mice. No behavioral effect after acute (nor sub-chronic) fluoxetine treatment was observed.
Our findings strengthen previous results demonstrating that chronic antidepressant treatment increases hippocampal neurogenesis in rodents. However, we could not correlate this to a behavioural outcome in the NSF test. Thus, the current data indicate the requirement for validated and stable methods in order to elucidate the functional significance of increased hippocampal neurogenesis.



TOP Unbiased estimation of the total number of NeuN positive neurons in
the developing neocortex

Thomas Krøigård, Lise Lyck, Nina Drøjdahl, and Bente Finsen
Medical Biotechnology Centre, University of Southern Denmark, Odense, Denmark


Stereology provides an unbiased and precise estimate of the total number of cells within a specific region.
In the investigation of neocortical development this technique offers an excellent means of quantifying the temporal changes in total cell number and changes in the number of neurons using cell specific markers. Neurons were visualized immunohistochemically using an antibody against NeuN, which is found in the nuclei of all neocortical neurons. NeuN positive neurons were counted in the neocortex of postnatal day 8 C57Bl6/J mice using thick (80 mm) vibratome sections cut in the saggital plane. Following mounting the sections had a mean thickness of 22.3 ± 2.6 mm (mean ± SD) which allowed us to use a 10 mm disector starting at 5 mm from the bottom of the section. Neocortex was defined as the neocortex proper, proisocortex, and periallocortex whereas allocortex and piriform cortex were excluded. Counting was performed in the right hemisphere which had been cut into five series yielding a section sampling fraction of 0.1. The area sampling fraction was 0.0008 based on a step length of 500 mm which gave a step area of 250,000 mm2 and the counting frame which had an area of 193 mm2. Counting six animals resulted in an estimate of 4.8 ± 0.5 (mean ± SD) million neurons. These data will be supplemented with estimates of the total number of NeuN positive neurons at postnatal days 0, 16, and in the adult mouse and estimates of total cell numbers in order to put this result into a developmental perspective.



TOP FRET FLIM microscopy
Jens R. Nyengaard1
Stereology and Electron Microscopy Research Laboratory, Institute of Clinical Medicine, University of Aarhus, Denmark


We are interested in “bridging” the gap between cellular and ultrastructural quantification to neurobiochemistry and neurophysiology by introducing two-photon excitation FRET (fluorescence resonance energy transfer) and FLIM (microscopy. Through advances in light microscopical technology, the ability to image specific protein molecules within neurobiological specimens will take basic neuroscience research to the next level. Historically neurobiology had been conducted at an impressive microscopic level. Through the utilization of clever methods for labeling brain areas of interest with standard staining protocols including immunohistochemistry, in-situ hybridization, fluorescent tagging, among others, great discoveries have been made. However, these discoveries inevitably lead to new questions. Interacting proteins assemble into molecular machines that control cellular homeostasis in living neurons. These protein assemblies were traditionally studied using biophysical or biochemical methods such as affinity chromatography or co-immunoprecipitation. While these in vitroscreening methods have the advantage of providing direct access to the genetic information encoding unknown protein partners, they do not however, allow direct access to interactions of these protein partners in their natural environment inside the living neuron. But using the approach of FRET/FLIM microscopy, this information can be obtained from single living neurons with nanometer resolution. However, many problems remain with 3- and 4-D quantification of the signals and mathematical manipulation of the spectral bleedthrough signal in two-photon FRET/FLIM microscopy.
With our interest and experience in microscopy and computer-assisted-stereological-toolbox microscopical systems as well as GFP mice we hope to foster an environment which would be ideal for the introduction of FRET/FLIM microscopy at Aarhus University.



TOP High sensation seeking men have increased dopamine release
in the right putamen during gambling.

J. Linnet; A. Gjedde; Y. Kumakura; P. Cumming; A. Møller*
PET-centre & CFIN, Aarhus University, Aarhus, Denmark


Sensation seeking is a personality trait based on Eysenck’s theory of optimal arousal, which has been associated with the dopaminergic system. High sensation seekers have a hedonic response to a higher level of stimulation, while low sensation seekers may react with aversion to the same level of stimulation. It is a common claim that high sensation seekers have a lower activity in the dopaminergic system which may make them susceptible for dopamine enhancing stimulants such as amphetamine and possibly gambling. This PET study focus on [11C]raclopride binding potential (pB) in high sensation seekers compared to low and mid-range sensation seekers in a control version and a gambling version of the Iowa Gambling Task. From a normally distributed sample of 243 individuals we defined cut-points of high and low sensation seekers as the top and bottom 20% of the distribution. This corresponded to a score of 25 and greater for high sensation seekers, 14 and lower for low sensation seekers, and 15 24 for mid-range sensation seeking. In the current study we compared 8 high sensation seeking men with 12 low to normal ranging sensation seeking men. Dynamic emission recordings were obtained during 60 minutes after i.v. [ C]raclopride (190 366 MBq) using the ECAT HR tomography. Maps of [ C]raclopride pB were calculated by the Logan reference tissue method with the cerebellum serving as reference and the mean pB calculated in templates for the putamen. High sensation seekers had a significantly lower [ C]raclopride binding potential in the right putamen (Mean SD: 3.0 0.1 vs. 2,9 0.1, p = 0.025), indicating increased dopamine occupancy of dopamine D2 and D3 receptors during the gambling session. No changes in the binding potential was observed in the normal/low sensation group. The increase in pB (contrast gamling task) in the right putamen was significantly larger in the high sensation seekers compared to normal/low sensation seekers (F = 5,74; p = 0,028) These preliminary results show increased dopamine release in the right putamen in high sensation seeking men while gambling.